PAR-2-IN-2
Product Specifications
CAS Number
313986-65-1
Target
Protease-activated Receptor, Serine Protease
Related Pathways
Proteases/Proteasome, GPCR/G Protein
Bioactivity
PAR-2-IN-2 (compound P-596) is an inhibitor of protease-activated receptor 2 (PAR-2), with an IC50 of 10.79 μM for SLIGKV and an IC50 greater than 200 μM for trypsin.
Smiles
O=C(C1=NN2C(N=C(C=C2C(F)(F)F)C=3C=CC=CC3)=C1)N4CCN(C(=O)C=5C=CC=CC5)CC4
Molecular Formula
C25H20F3N5O2
Molecular Weight
479.454
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog