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PF-06422913

Product Specifications

CAS Number

1539296-46-2

Target

GluR

Related Pathways

Neuroscience

Bioactivity

PF-06422913 is an orally active, potent, and selective negative allosteric modulator of the metabotropic glutamate receptor 5 (mGluR5) .

Smiles

FC(F)(F)C=1C=CN=CC1C2=NN(C=3N=C(OCC4=NC=CC=C4)C=NC23)C

Molecular Formula

C18H13F3N6O

Molecular Weight

386.331

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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