TRF2-IN-1
Product Specifications
Target
Telomerase, Apoptosis
Related Pathways
DNA Damage/DNA Repair, Apoptosis
Bioactivity
TRF2-IN-1 (compound F2) is a potent inhibitor of telomere repeat-binding factor 2 (TRF2) . It exhibits antiproliferative activity and induces apoptosis. TRF2-IN-1 binds directly to the TRF2TRFH domain, selectively inhibiting TRF2 protein expression and telomere localization. Additionally, TRF2-IN-1 possesses anticancer properties and shows potential for osteosarcoma research.
Smiles
COC1=CC(=C(C(=C1)OC)C(=O)/C=C/C2=CC(=CC=C2)Br)OC
Molecular Formula
C18H17BrO4
Molecular Weight
377.229
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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