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TRF2-IN-1

Product Specifications

Target

Telomerase, Apoptosis

Related Pathways

DNA Damage/DNA Repair, Apoptosis

Bioactivity

TRF2-IN-1 (compound F2) is a potent inhibitor of telomere repeat-binding factor 2 (TRF2) . It exhibits antiproliferative activity and induces apoptosis. TRF2-IN-1 binds directly to the TRF2TRFH domain, selectively inhibiting TRF2 protein expression and telomere localization. Additionally, TRF2-IN-1 possesses anticancer properties and shows potential for osteosarcoma research.

Smiles

COC1=CC(=C(C(=C1)OC)C(=O)/C=C/C2=CC(=CC=C2)Br)OC

Molecular Formula

C18H17BrO4

Molecular Weight

377.229

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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