CDK2/9-IN-1
Product Specifications
CAS Number
2222285-23-4
Target
Apoptosis, CDK
Related Pathways
Apoptosis, Cell Cycle/Checkpoint
Bioactivity
CDK2/9-IN-1 (compound 20a) is an orally active dual inhibitor of CDK2 and CDK9, with IC50 values of 0.004 μM and 0.009 μM for CDK2 and CDK9, respectively. It induces apoptosis by regulating G2/M cell cycle arrest and exhibits antitumor activity.
Smiles
O=S(=O)(N)C1=CC=C(C=C1)NC2=NC=C(C(=N2)NC3=NC=CS3)C
Molecular Formula
C14H14N6O2S2
Molecular Weight
362.43
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
P1001-31C1 50 µg
P53 DINP1 (p53 Dependent Damage-inducible Nuclear Protein, SIP, Stress Induced Protein) discontinued
Sign In for Pricing
View Details