What is the catalog number for PKMYT1-IN-8?

The catalog number for PKMYT1-IN-8 is T204125.

What sizes are available for PKMYT1-IN-8?

PKMYT1-IN-8 is available in the following size(s): 10 mg, 50 mg.

How many pack sizes does PKMYT1-IN-8 come in?

PKMYT1-IN-8 is available in 2 different pack sizes.

Is PKMYT1-IN-8 in stock?

PKMYT1-IN-8 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures PKMYT1-IN-8?

PKMYT1-IN-8 is manufactured by Molfinity.

What is the estimated delivery time for PKMYT1-IN-8?

Estimated delivery time for PKMYT1-IN-8 is approximately 10 business day(s), depending on your location.

PKMYT1-IN-8

Product Specifications

Target

Ephrin Receptor, Wee1

Related Pathways

Tyrosine Kinase/Adaptors, Cell Cycle/Checkpoint

Bioactivity

PKMYT1-IN-8 (Compound 137) is an inhibitor of PKMYT1, with an IC50 value of 9 nM. It also inhibits EPHB3, EPHA1, KIT, EPHB1, EPHA2, EPHA3, and EPHB2, exhibiting IC50 values of 1.79, 3.17, 4.29, 6.32, 6.83, 8.10, and 10.9 μM, respectively. Additionally, PKMYT1-IN-8 suppresses the proliferation of cancer cells OVCAR3 with a GI50 of 2.02 μM.