PF-4363467
Product Specifications
CAS Number
2040055-84-1
Target
Dopamine Receptor
Related Pathways
GPCR/G Protein, Neuroscience
Bioactivity
PF-4363467 is a dopamine D3/D2 receptor antagonist that reduces opioid-seeking behavior without the side effects associated with D2 receptors. It has a Ki value of 3.1 nM for D3R and 692 nM for D2R.
Smiles
CC=1C=C(C=CC1NS(=O)(=O)C2=CC=C(C(C)C)C=C2)[C@@H]3CN(CC)CCO3
Molecular Formula
C22H30N2O3S
Molecular Weight
402.55
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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