KOR agonist 3
Product Specifications
Target
Opioid Receptor
Related Pathways
Neuroscience, Endocrinology/Hormones, GPCR/G Protein
Bioactivity
KOR agonist 3 (Compound 5) is an agonist of the κ opioid receptor (κOR) with an EC50 of 0.88 nM. It also exhibits some activation of μOR, with an EC50 of 720 nM. However, KOR agonist 3 does not activate δOR at concentrations below 1 μM. Its ability to recruit β-Arrestin-2 is lower than that of U50488.
Molecular Formula
C24H24N2O3
Molecular Weight
388.46
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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