SR-12062
Product Specifications
CAS Number
1623019-77-1
Bioactivity
SR-12062 functions as a full agonist at neurotensin receptor 1 (NTSR1), demonstrating notable efficacy and increased potency. Its EC50 value on NTSR1 is 2 μM, with complete receptor activation (Emax=100%) . Compared to the parent compound 1 (EC50=178 μM; Emax=17%), SR-12062 shows approximately 90-fold greater potency.
Smiles
C(C(N[C@@H](CC(C)C)C(O)=O)=O)N1C=2C(=CC(=CC2)C3=CC4=C(N=C3)C=CC=C4)C=C1
Molecular Formula
C25H25N3O3
Molecular Weight
415.48
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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