Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

PF-03654764 tosylate

Product Specifications

CAS Number

1337536-85-2

Bioactivity

PF-03654764 exhibits high affinity for the human H3 receptor, but displays significantly lower affinity for the rat H3 receptor, with over 1000-fold selectivity against other human histamine receptor subtypes (H1, H2, and H4) . In functional assays measuring cAMP using reporter gene assays (β-lactamase) conducted in HEK293 cells stably expressing the full-length human or rat H3 receptor, PF-03654764 demonstrated potent antagonist properties.

Smiles

S(=O)(=O)(O)C1=CC=C(C)C=C1.F[C@@]1(C[C@@H](C(NCC(C)C)=O)C1)C2=CC(F)=C(CN3CCCC3)C=C2

Molecular Formula

C20H28F2N2O xC7H8O3S

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Mouse Monoclonal Feline Immunodeficiency Virus Antibody (NM3-6A9) [Alexa Fluor 594]
NB100-66500AF594 0.1 mL

Mouse Monoclonal Feline Immunodeficiency Virus Antibody (NM3-6A9) [Alexa Fluor 594]

Sign In for Pricing
View Details
rno-miR-499 Primers
MP-r00204 150 µL - 10 µM

rno-miR-499 Primers

Sign In for Pricing
View Details
Research Grade Onfekafusp Alfa
DHK09501 100 μg

Research Grade Onfekafusp Alfa

Sign In for Pricing
View Details
GAD1/2 antibody
70R-49776 100 ul

GAD1/2 antibody

Sign In for Pricing
View Details
PANK1/2 (C-4) PE
sc-390595 PE 200 µg/mL

PANK1/2 (C-4) PE

Sign In for Pricing
View Details
MYBPC3 Mouse Monoclonal Antibody [Clone 2D8D7]
E45M21268V-2 50 µL

MYBPC3 Mouse Monoclonal Antibody [Clone 2D8D7]

Sign In for Pricing
View Details