Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

PF-03654764 tosylate

Product Specifications

CAS Number

1337536-85-2

Bioactivity

PF-03654764 exhibits high affinity for the human H3 receptor, but displays significantly lower affinity for the rat H3 receptor, with over 1000-fold selectivity against other human histamine receptor subtypes (H1, H2, and H4) . In functional assays measuring cAMP using reporter gene assays (?-lactamase) conducted in HEK293 cells stably expressing the full-length human or rat H3 receptor, PF-03654764 demonstrated potent antagonist properties.

Smiles

S(=O)(=O)(O)C1=CC=C(C)C=C1.F[C@@]1(C[C@@H](C(NCC(C)C)=O)C1)C2=CC(F)=C(CN3CCCC3)C=C2

Molecular Formula

C20H28F2N2O xC7H8O3S

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

Explore Other Products

Discover premium biology products from our extensive collection of 20M+ items

Mouse Pcm1 Pre-designed siRNA Set B

SI110231B 1 Each

Mouse Pcm1 Pre-designed siRNA Set B

Ask

DGKA Mouse Monoclonal Antibody (Biotin conjugated) [Clone ID: OTI3G7]

TA504024AM 100 µL

DGKA Mouse Monoclonal Antibody (Biotin conjugated) [Clone ID: OTI3G7]

Ask

GPSM3 discontinued

536956-01 30ul

GPSM3 discontinued

Ask

GPSM3 discontinued

536956-02 100 µL

GPSM3 discontinued

Ask

Recombinant Human CCS/SOD4 Protein

NBP1-48393-0.5mg 0.5 mg

Recombinant Human CCS/SOD4 Protein

Ask

NADK2 Knockout MES-OV Polyclonal Cells

ARG6186 1 Million

NADK2 Knockout MES-OV Polyclonal Cells

Ask