Gintemetostat
Product Specifications
CAS Number
2604513-16-6
Target
Histone Methyltransferase
Related Pathways
Chromatin/Epigenetic
Bioactivity
Gintemetostat (KTX-1001) is a potent and selective small molecule inhibitor of nuclear receptor-binding SET domain protein 2 (NSD2), exhibiting IC50 values ranging from 0.001 μM to 0.01 μM, and it belongs to the chemical class of piperidinyl-methyl-purineamine derivatives, with primary research applications in oncology for the treatment of NSD2-dysregulated cancers.
Smiles
C(C=1C(=CN=C(C1)C2=C(F)C=C(OC)C(F)=C2)N3C[C@]([C@@H](C(F)F)O)(N)CCC3)N4C=5C(N=C4)=C(N)N=CN5
Molecular Formula
C25H26F4N8O2
Molecular Weight
546.52
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
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