What is the catalog number for Flucopride?

The catalog number for Flucopride is T201815.

What sizes are available for Flucopride?

Flucopride is available in the following size(s): 10 mg, 50 mg.

How many pack sizes does Flucopride come in?

Flucopride is available in 2 different pack sizes.

Is Flucopride in stock?

Flucopride is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures Flucopride?

Flucopride is manufactured by Molfinity.

What is the estimated delivery time for Flucopride?

Estimated delivery time for Flucopride is approximately 10 business day(s), depending on your location.

Flucopride

Product Specifications

CAS Number

1639925-34-0

Target

Cholinesterase (ChE), 5-HT Receptor

Related Pathways

GPCR/G Protein, Neuroscience

Bioactivity

Flucopride (Compound 4a) acts as an acetylcholinesterase inhibitor (AChE) with an IC50 value of 24 nM and serves as a partial agonist for the human 5-HT4 receptor (5-HT4R) with a Ki of 9.6 nM for (h) 5-HT4R. It promotes non-amyloidogenic processing of APP in COS-7 cells transiently expressing (h) 5-HT4R with an EC50 of 23.0 nM. Flucopride is also likely to exhibit significant gastrointestinal tract (GIT) penetration and blood-brain barrier (BBB) permeability, as determined in PAMPA experiments.