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ATR kinase-IN-3

Product Specifications

CAS Number

1613196-92-1

Target

ATM/ATR

Related Pathways

PI3K/Akt/mTOR signaling|||DNA Damage/DNA Repair

Bioactivity

ATRkinase-IN-3 (Compound I-G-28) is an inhibitor of the ATR protein kinase, exhibiting a Ki value ranging from 0.01 to 1 ?M, and is utilized in cancer research.

Smiles

O=C(NC=1C=NC=C(F)C1N2CCC(C(=O)N3CCNC4(C3)CC4)CC2)C=5C(=NN6C=C(F)C=NC56)N

Molecular Formula

C24H27F2N9O2

Molecular Weight

511.53

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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