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L134

Product Specifications

Target

PROTACs|||Epigenetic Reader Domain

Related Pathways

Chromatin/Epigenetic|||PROTAC

Bioactivity

L134, an effective PROTAC BRD4 degrader, exhibits a DC50 value of 7.36 nM. The degradation of BRD4 by L134 is mediated through the ubiquitin-proteasome system in a DCAF11-dependent manner.

Molecular Formula

C48H51ClF3N7O7S

Molecular Weight

962.47

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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