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ETP-45835 dihydrochloride

Product Specifications

CAS Number

2136571-30-5

Target

TLR, ERK

Related Pathways

MAPK, Immunology/Inflammation

Bioactivity

D-106669, an inhibitor of Erk2, exhibits an IC50 of 18.7 μM and effectively suppresses cell proliferation with an EC50 of 0.9 μM.

Smiles

C1(C2=NNC(C3CCNCC3)=C2)=CC=NC=C1.Cl.Cl

Molecular Formula

C13H18Cl2N4

Molecular Weight

301.22

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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