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SJ1008066

Product Specifications

CAS Number

2758867-71-7

Target

Androgen Receptor|||FGFR

Related Pathways

Endocrinology/Hormones|||Tyrosine Kinase/Adaptors|||Angiogenesis

Bioactivity

SJ1008066 is a MAGE-A11 inhibitor with an IC50 of 0.13 ?M. It binds to the MAGE homology domain (MHD) and disrupts the MAGE-A11:PCF11 interaction.

Smiles

N=1C=CC(NCCCNCC=2C=CC=3NC=CC3C2)=C4C=CC=CC14

Molecular Formula

C21H22N4

Molecular Weight

330.43

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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