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NMDAR antagonist 2

Product Specifications

Target

IGluR

Related Pathways

Membrane transporter/Ion channel|||Neuroscience

Bioactivity

NMDAR antagonist 2 (compound 3I) is a blood-brain barrier permeable antagonist of NMDA receptors, exhibiting IC50 values of 4.42 ?M and 214.75 ?M at membrane potentials of -60 mV and 40 mV, respectively, for hGluN1/hGluN2A. This compound has been shown to mitigate hippocampal damage.

Molecular Formula

C17H20ClNO

Molecular Weight

289.8

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Product Datasheet

https://www.targetmol.com/attachment/DataSheet/274139177807773858/T201550

Available Sizes

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