PROTAC BRM/BRG1 degrader-2
Product Specifications
CAS Number
2933124-32-2
Target
Epigenetic Reader Domain|||PROTACs
Related Pathways
PROTAC|||Chromatin/Epigenetic
Bioactivity
PROTAC BRM/BRG1 degrader-2 (Example.004) is a potent PROTAC BRM/BRG1 degrading agent exhibiting a DC50 of less than 10 nM and an IC50 of 15 nM in A549 cells.
Smiles
NC=1C=2C(N(N1)C3CCN(CC3)C=4N=CC(=CN4)[C@H]5CC[C@H](C(N[C@H](C(=O)N6[C@H](C(N[C@@H](C)C7=CC=C(C=C7)C8=C(C)N=CS8)=O)C[C@@H](O)C6)[C@@](C)(C)C)=O)CC5)=CC(=NN2)C9=C(O)C=CC=C9
Molecular Formula
C50H60N12O5S
Molecular Weight
941.15
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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