What is the catalog number for EGFR-IN-131?

The catalog number for EGFR-IN-131 is T201154.

What sizes are available for EGFR-IN-131?

EGFR-IN-131 is available in the following size(s): 10 mg, 50 mg.

How many pack sizes does EGFR-IN-131 come in?

EGFR-IN-131 is available in 2 different pack sizes.

Is EGFR-IN-131 in stock?

EGFR-IN-131 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures EGFR-IN-131?

EGFR-IN-131 is manufactured by Molfinity.

What is the estimated delivery time for EGFR-IN-131?

Estimated delivery time for EGFR-IN-131 is approximately 10 business day(s), depending on your location.

EGFR-IN-131

Product Specifications

Target

Apoptosis, EGFR

Related Pathways

Tyrosine Kinase/Adaptors, JAK/STAT signaling, Angiogenesis, Apoptosis

Bioactivity

EGFR-IN-131 (compound 3a) is an efficacious EGFR inhibitor capable of crossing the blood-brain barrier, with an IC50 value of 272.9 nM. This compound exhibits anti-proliferative activity, induces cellular apoptosis (apoptosis), and causes cell cycle arrest in the G0/G1 phase. Additionally, EGFR-IN-131 reduces the protein expression of p-EGFR.

Smiles

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