RET-IN-27
Product Specifications
Target
C-RET
Related Pathways
Tyrosine Kinase/Adaptors, Apoptosis
Bioactivity
RET-IN-27 (compound 20p) serves as a potent inhibitor of RET, exhibiting IC50 values of 3.6 nM for RETWT, 0.1 nM for RETV804L, 2.1 nM for RETV804M, and 0.3 nM for RETM918T. This compound plays a significant role in cancer research.
Molecular Formula
C31H28N8O
Molecular Weight
528.61
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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