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RET-IN-27

Product Specifications

Target

C-RET

Related Pathways

Tyrosine Kinase/Adaptors|||Apoptosis

Bioactivity

RET-IN-27 (compound 20p) serves as a potent inhibitor of RET, exhibiting IC50 values of 3.6 nM for RETWT, 0.1 nM for RETV804L, 2.1 nM for RETV804M, and 0.3 nM for RETM918T. This compound plays a significant role in cancer research.

Molecular Formula

C31H28N8O

Molecular Weight

528.61

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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