PROTAC BRM/BRG1 degrader-4
Product Specifications
Target
PROTACs, Epigenetic Reader Domain
Related Pathways
Chromatin/Epigenetic, PROTAC
Bioactivity
PROTAC BRM/BRG1 degrader-4 (example 047) is a potent degrader targeting both BRM and BRG1, demonstrating DC50 values of 0.21 nM and 3.4 nM respectively in SW1573 cells.
Smiles
N#CC=1C=C2N=C(NC2=C(OC)C1)C3=C(N=CC(C4=CC(F)=CC(=C4)C)=C3N5CCC(N)CC5)N
Molecular Formula
C44H52N10O6S
Molecular Weight
849.01
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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