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Keap1-Nrf2-IN-24

Product Specifications

Target

Nrf2

Related Pathways

Immunology/Inflammation

Bioactivity

Keap1-Nrf2-IN-24 (compound 57) is an effective Keap1-Nrf2 inhibitor with a Ki value of 13 nM. This compound enhances the protein expression of TRXR1 and NQO1, as well as the mRNA expression of AKR1B10. Additionally, Keap1-Nrf2-IN-24 demonstrates good metabolic stability.

Molecular Formula

C32H25FN4O5S

Molecular Weight

596.63

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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