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IMPDH2-IN-4

Product Specifications

Target

VEGFR, CDK

Related Pathways

Angiogenesis, Tyrosine Kinase/Adaptors, Cell Cycle/Checkpoint

Bioactivity

IMPDH2-IN-4 (compound 2d) is a Mycophenolic acid analog and a selective IMPDH2 inhibitor with a Ki of 1.8 μM. It exhibits potent cytotoxic activity against osteosarcoma cancer cell lines. Additionally, IMPDH2-IN-4 demonstrates high affinity for VEGFR-2, CDK2, and IMPDH.

Molecular Formula

C35H34O6Si

Molecular Weight

578.73

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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