STING-IN-10
Product Specifications
Target
PROTACs, STING
Related Pathways
PROTAC, Immunology/Inflammation
Bioactivity
STING-IN-10 (P8) serves as both a dual degrader and inhibitor of STING, exhibiting an impressive DC50 value of 2.58 μM in THP-1 cells. This compound also demonstrates anti-inflammatory activity.
Smiles
O=C(N)C(N(C1=NC(N)=C(S1)C(=O)C2=CC=C(C=C2)S(F)(F)(F)(F)F)C3=CC=C(F)C=C3)C
Molecular Formula
C35H33N7O11
Molecular Weight
727.68
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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