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DS06652923

Product Specifications

Target

EGFR

Related Pathways

Tyrosine Kinase/Adaptors|||JAK/STAT signaling|||Angiogenesis

Bioactivity

DS06652923 is an orally active inhibitor targeting EGFR triple mutations. It exhibits growth-inhibitory effects on Ba/F3EGFRdel19/T90M/C795S cells, with a GI50 value of 9.4 nM. Additionally, DS06652923 induces tumor regression in the Ba/F3 syngeneic transplantation model.

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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