FLT3/HDAC-IN-1
Product Specifications
Target
Apoptosis, FLT, HDAC
Related Pathways
Tyrosine Kinase/Adaptors, Apoptosis, Chromatin/Epigenetic, DNA Damage/DNA Repair, Angiogenesis
Bioactivity
FLT3/HDAC-IN-1 is a dual inhibitor targeting FLT3 and HDAC, with IC50 values of 30.4 nM for FLT3 and 52.4, 14.7 nM for HDAC1/3, respectively. It induces apoptosis in MV-4-11 cells and exhibits antiproliferative effects against BaF3 cells transformed by FLT3 mutations. FLT3/HDAC-IN-1 is useful for research on refractory solid tumors and hematological malignancies.
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog