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STAT3-IN-34

Product Specifications

Target

STAT

Related Pathways

Stem Cells, JAK/STAT signaling

Bioactivity

STAT3-IN-34 (Compound 15E) acts as a STAT3 inhibitor, blocking both the nuclear translocation and the transcriptional regulator activity of STAT3. It effectively inhibits HaCaT cell proliferation with an IC50 value of 0.008 μM. Additionally, STAT3-IN-34 reduces IL-17A expression and mitigates Imiquimod-induced psoriasis in mouse models.

Molecular Formula

C19H16N2O4S

Molecular Weight

368.41

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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