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HIV-1 inhibitor-75

Product Specifications

Target

Reverse Transcriptase|||HIV Protease

Related Pathways

Proteases/Proteasome|||Microbiology/Virology

Bioactivity

HIV-1inhibitor-75 is a human immunodeficiency virus 1 (HIV-1) inhibitor with an EC50 range of 0.0039-0.338 ?M. Its target is the reverse transcriptase, exhibiting an IC50 value of 0.055 ?M. Additionally, HIV-1inhibitor-75 demonstrates good metabolic stability in vitro, presenting moderate clearance rates and an extended half-life in human plasma and liver microsomes.

Molecular Formula

C25H20ClN3O3S

Molecular Weight

477.96

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

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