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ONCOII

Product Specifications

CAS Number

1263564-94-8

Target

Kinesin

Related Pathways

Cytoskeletal Signaling

Bioactivity

ONCOII, an inhibitor of Mps1 with an IC50 of 10.8 nM, exhibits varying inhibitory activities depending on naturally occurring mutations within the Mps1 gene. Cells harboring Mps1 mutations demonstrate increased resistance to ONCOII. This compound is applicable in cancer research.

Smiles

N#CC1=CC=C(N=C1NC2CCCCC2)NC=3C=CC(=C(OCC#N)C3)C=4C=NN(C4)C

Molecular Formula

C24H25N7O

Molecular Weight

427.5

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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