VEGFR-2/InhA-IN-1
Product Specifications
Target
VEGFR, Antibacterial
Related Pathways
Angiogenesis, Tyrosine Kinase/Adaptors, Microbiology/Virology
Bioactivity
VEGFR-2/InhA-IN-1, a dual inhibitor based on pyrazole, targets InhA and VEGFR, exhibiting both anti-tuberculosis and anti-angiogenic properties. It demonstrates effective antibacterial activity against the Mycobacterium tuberculosis H37Rv strain (MIC = 6.25 μg/mL) and significantly suppresses VEGFR-2 activity (IC 50 = 15.27 nM) .
Molecular Formula
C22H16ClFN4O
Molecular Weight
406.84
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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