(2R,3S) -Azelaprag
Product Specifications
CAS Number
2049979-31-7
Target
Apelin receptor
Related Pathways
GPCR/G Protein
Purity
>99.99%
Bioactivity
(2R,3S) -N- (4- (2,6-dimethoxyphenyl) -5- (5-methylpyridin-3-yl) -4H-1,2,4-triazol-3-yl) -3- (5-methylpyrimidin-2-yl) butane-2-sulfonamide is an Apelin receptor agonist with an EC50 for Apelin receptors of 0.012 μM. (2R,3S) -N- (4- (2,6-dimethoxyphenyl) -5- (5-methylpyridin-3-yl) -4H-1,2,4-triazol-3-yl) -3- (5- methylpyrimidin-2-yl) butane-2-sulfonamide is used in the treatment of heart failure, atherosclerosis, obesity, diabetes mellitus, amyotrophic lateral sclerosis, coronary artery disease, hypertension, stroke and myocardial infarction.
Smiles
N(S([C@@H]([C@@H](C)C=1N=CC(C)=CN1)C)(=O)=O)C=2N(C(=NN2)C=3C=C(C)C=NC3)C4=C(OC)C=CC=C4OC
Molecular Formula
C25H29N7O4S
Molecular Weight
523.61
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
302412-ML550 100 µL
Ehmt2 (Histone-lysine N-Methyltransferase EHMT2, 211-, Euchromatic Histone-lysine N-Methyltransferase 2, HLA-B-Associated Transcript 8, Histone H3-K9 Methyltransferase 3, H3-K9-HMTase 3, Protein G9a, Ehmt2, Bat8, G9a, Ng36) (MaxLight 550) discontinued
Sign In for Pricing
View Details