(2R,3S) -Azelaprag
Product Specifications
CAS Number
2049979-31-7
Target
Apelin receptor
Related Pathways
GPCR/G Protein
Purity
>99.99%
Bioactivity
(2R,3S) -N- (4- (2,6-dimethoxyphenyl) -5- (5-methylpyridin-3-yl) -4H-1,2,4-triazol-3-yl) -3- (5-methylpyrimidin-2-yl) butane-2-sulfonamide is an Apelin receptor agonist with an EC50 for Apelin receptors of 0.012 μM. (2R,3S) -N- (4- (2,6-dimethoxyphenyl) -5- (5-methylpyridin-3-yl) -4H-1,2,4-triazol-3-yl) -3- (5- methylpyrimidin-2-yl) butane-2-sulfonamide is used in the treatment of heart failure, atherosclerosis, obesity, diabetes mellitus, amyotrophic lateral sclerosis, coronary artery disease, hypertension, stroke and myocardial infarction.
Smiles
N(S([C@@H]([C@@H](C)C=1N=CC(C)=CN1)C)(=O)=O)C=2N(C(=NN2)C=3C=C(C)C=NC3)C4=C(OC)C=CC=C4OC
Molecular Formula
C25H29N7O4S
Molecular Weight
523.61
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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