NF-56-EJ40 hydrochloride
Product Specifications
CAS Number
2728500-80-7
Target
Succinate Receptor 1 (SUCNR1)
Related Pathways
GPCR/G Protein
Purity
0.9933
Bioactivity
NF-56-EJ40 hydrochloride is a potent, high-affinity, and highly selective human SUCNR1 (GPR91) antagonist with an IC50 of 25 nM and a Ki of 33 nM, and shows almost no activity towards rat SUCNR1. NF-56-EJ40 hydrochloride has high affinity for humanized rat SUCNR1 with a Ki value of 17.4 nM.
Smiles
O=C(CC1=C(NC(C2=CC=CC(C3=CC=C(CN4CCN(CC4)C)C=C3)=C2)=O)C=CC=C1)O.Cl.Cl
Molecular Formula
C27H31Cl2N3O3
Molecular Weight
516.46
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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