Amastatin
Amastatin is A slow, tightly bound, competitive inhibitor of aminopeptidase (AP) with an IC50 of 0.54 μg/mL for AP-A[1][2].
Product Specifications
CAS Number
67655-94-1
UNSPSC
12352211
Hazard Statement
H315-H319-H335
Target
Aminopeptidase
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/amastatin.html
Solubility
10 mM in DMSO
Smiles
O=C(C[C@H](NC([C@@H](NC([C@@H](NC([C@H]([C@@H](CC(C)C)N)O)=O)C(C)C)=O)C(C)C)=O)C(O)=O)O
Molecular Formula
C21H38N4O8
Molecular Weight
474.55
Precautions
P261-P264-P271-P280-P302+P352-P304+P340-P305+P351+P338-P362+P364-P403+P233-P405-P501
References & Citations
[1]Aoyagi T, et al. Amastatin, an inhibitor of aminopeptidase A, produced by actinomycetes. J Antibiot (Tokyo) . 1978 Jun;31 (6) :636-8.|[2]Wilkes SH, et al. The slow, tight binding of bestatin and amastatin to aminopeptidases. J Biol Chem. 1985 Oct 25;260 (24) :13154-62.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
N000153 30 Pack (30 Marker (s) x 1 Roll)
Nitr.desod.450x52RL-T1-LL-P21 Pipe Markers for Acids & Bases
Sign In for Pricing
View Details