Amastatin
Amastatin is A slow, tightly bound, competitive inhibitor of aminopeptidase (AP) with an IC50 of 0.54 μg/mL for AP-A[1][2].
Product Specifications
CAS Number
67655-94-1
UNSPSC
12352211
Hazard Statement
H315-H319-H335
Target
Aminopeptidase
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/amastatin.html
Solubility
10 mM in DMSO
Smiles
O=C(C[C@H](NC([C@@H](NC([C@@H](NC([C@H]([C@@H](CC(C)C)N)O)=O)C(C)C)=O)C(C)C)=O)C(O)=O)O
Molecular Formula
C21H38N4O8
Molecular Weight
474.55
Precautions
P261-P264-P271-P280-P302+P352-P304+P340-P305+P351+P338-P362+P364-P403+P233-P405-P501
References & Citations
[1]Aoyagi T, et al. Amastatin, an inhibitor of aminopeptidase A, produced by actinomycetes. J Antibiot (Tokyo) . 1978 Jun;31 (6) :636-8.|[2]Wilkes SH, et al. The slow, tight binding of bestatin and amastatin to aminopeptidases. J Biol Chem. 1985 Oct 25;260 (24) :13154-62.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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