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VU0810464

Product Specifications

Background

VU0810464 is potent (Kir3.1/3.2; GIRK1/2 EC50 = 165 nM) activator of G protein-gated inwardly-rectifying potassium channels (Kir3; GIRK) .1,2 Displays selectivity for Kir3.1/3.2 versus Kir3.1/3.4 as well as selectivity for neuronal versus cardiac Kir3 channels. VU0810464 reduced stress-induced hyperthermia but not anxiety-related behavior in mice.

Conjugation

Unconjugated

Buffer

White solid

Storage Conditions

-20°C

Available Sizes

Frequently Asked Questions

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