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Fulvestrant

Product Specifications

Background

A 17β-estradiol analog that acts as an estrogen receptor (ER) antagonist and GPR30/GPER agonist with high binding affinity.1,2 First-in-class SERD (selective ER degrader) because it inhibits ER transcriptional activity and leads to its degradation.3 Exhibits mixed neuroprotective activity in vivo.4 Clinically useful option for some advanced breast cancers.5

Conjugation

Unconjugated

Buffer

White solid

Storage Conditions

-20°C

Available Sizes

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