Fulvestrant
Product Specifications
Background
A 17β-estradiol analog that acts as an estrogen receptor (ER) antagonist and GPR30/GPER agonist with high binding affinity.1,2 First-in-class SERD (selective ER degrader) because it inhibits ER transcriptional activity and leads to its degradation.3 Exhibits mixed neuroprotective activity in vivo.4 Clinically useful option for some advanced breast cancers.5
Conjugation
Unconjugated
Buffer
White solid
Storage Conditions
-20°C
Available Sizes
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