What is the catalog number for CPI203?

The catalog number for CPI203 is bs-82778C.

What sizes are available for CPI203?

CPI203 is available in the following size(s): 5 mg, 25 mg.

How many pack sizes does CPI203 come in?

CPI203 is available in 2 different pack sizes.

CPI203 is currently made to order / not held in immediate stock. Contact us for lead time.

CPI203

Product Specifications

Background

CPI203, a JQ1 analog, is a potent and selective inhibitor of the BET bromodomain BRD4 (IC50 = 26 nM) .1 It helps promote the maintenance of hematopoietic stem cells via repression of Myc expression.2 CPI203 reversibly suppressed intestinal stem cell differentiation in a mouse model.3 It enhanced the expansion of human cord blood hematopoietic stem cells without losing cell viability.4 CPI203 displays synergistic antitumor activity with various agents including lenalidomide5, bortezomib6, and PARP inhibitors7.