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EPZ015666

Product Specifications

Background

EPZ015666 is a selective and potent (IC50 = 22nM) inhibitor of arginine methyltransferase 5 (PRMT5) .1,2 PRMT5 inhibition with EPZ015666 potently suppressed in vivo glioblastoma tumors3 and significantly inhibited the growth of multiple myeloma cell lines4.

Conjugation

Unconjugated

Buffer

White solid

Storage Conditions

-20°C

Product Datasheet

https://www.biossantibodies.com/datasheets/bs-82770C

Available Sizes

Curated Selection

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