PF-05089771
Product Specifications
Background
Potent and selective inhibitor of the voltage gated sodium channel 1.7 (Nav1.7) .1,3 It is a state-dependent inhibitor with IC50 = 11 nM for the half-inactivated channels and IC50 ~ 10 µM for resting channels.1 Equipotent for human, monkey, dog, and mouse channels but 15x less potent for rat channels. Interacts equally with fast and slow inactivated Nav1.7 channels.2
Conjugation
Unconjugated
Buffer
White solid
Storage Conditions
-20°C
Available Sizes
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