Cilostamide
Product Specifications
Background
Selective inhibitor of phosphodiesterase-3 (PDE3) . Displays limited selectivity for PDE3A versus PDE3B (IC50 = 27 and 50 nM) 1,2. Blocks PKB/Akt signaling pathway downstream via inhibition of Akt-activated PDE3B3. Reverses the effect of leptin on food intake and body weight4.
Conjugation
Unconjugated
Buffer
White solid
Storage Conditions
RT
Available Sizes
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