Bupropion HCl
Product Specifications
Background
Clinically useful antidepressant that inhibits monoamine transporters DAT, NET, and SERT (Kis for dopamine uptake = 2.8, 1.4, 45 µM) .1 Also acts as a noncompetitive antagonist at nicotinic acetylcholine receptors (AChRs) .2 At higher concentrations (50 µM), stimulates pro-inflammatory cytokines and TLR2/TLR4 and JAK2/STAT3 in human peripheral blood mononuclear cells (PBMCs) .3
Conjugation
Unconjugated
Buffer
White solid
Storage Conditions
-20°C
Available Sizes
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