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Pranlukast

Product Specifications

Background

Pranlukast is a selective Leukotriene CysLT1 antagonist1 and has been used in the treatment of asthma2. Pranlukast is also an inhibitor of GPR173 (IC50’s = 10.5nM hGPR17, 31nM rGPR17) and is superior to Montelukast in achieving functional inhibition4.

Conjugation

Unconjugated

Buffer

White solid

Storage Conditions

RT

Available Sizes

Frequently Asked Questions

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