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Zebularine

Product Specifications

Background

Orally active DNA methyltransferase inhibitor. Inhibits tumor cell proliferation (IC50 = 120 μM) and re-activates silenced genes in T24 bladder carcinoma cells. Inhibits cytidine deaminase (Ki ~ 2 μM) ; induces differentiation of mesenchymal stem cells into cardiomyocytes.

Conjugation

Unconjugated

Buffer

White solid

Storage Conditions

-20°C

Available Sizes

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