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GDC-0941

Product Specifications

Background

GDC-0941 is a potent and selective inhibitor of class I phosphatidylinositol-3-kinases (PI3K) with significant antitumor activity – IC50’s: PI3Kα = 3nM, PI3Kβ = 33 nM, PI3Kδ = 3 nM, PI3Kγ = 75 nM.1,2 GDC-0941 is the chemical probe of choice for the pan-inhibition of class I PI3K’s.3 Currently in clinical trials.4

Conjugation

Unconjugated

Buffer

Solid

Storage Conditions

-20°C

Product Datasheet

https://www.biossantibodies.com/datasheets/bs-82409C

Available Sizes

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