What is the catalog number for Enzastaurin?

The catalog number for Enzastaurin is bs-82405C.

What sizes are available for Enzastaurin?

Enzastaurin is available in the following size(s): 5 mg, 25 mg.

How many pack sizes does Enzastaurin come in?

Enzastaurin is available in 2 different pack sizes.

Is Enzastaurin in stock?

Enzastaurin is currently made to order / not held in immediate stock. Contact us for lead time.

Enzastaurin

Product Specifications

Background

Potent and selective PKCβ inhibitor. IC50 = 6, 39, 83 and 110 nM, for PKCβ, PKCα, PKCγ and PKCε respectively.1 Induces apoptosis in multiple myeloma cell lines via inhibition of the AKT signaling pathway.2 Induces mitotic missegregation and preferential cytotoxicity in colorectal cancer cells with chromosomal instability.3 Attenuates ampheta-mine-stimulated dopamine efflux.4 Inhibits blood-brain barrier leakiness in a mouse model.5