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TGN-020

Product Specifications

Background

Aquaporin 4 channel blocker, IC50 = 3.1 μM.1 Reduces ischemic cerebral edema in a mouse model of focal cerebral ischemia using MRI.2 Increases regional cerebral blood flow as determined in wild-type and AQP-4 knockout mice.3 Reduces brain edema when administered after onset of ischemia in rat models.4

Conjugation

Unconjugated

Buffer

Off-white solid

Storage Conditions

RT

Available Sizes

Frequently Asked Questions

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